首页> 外文OA文献 >Aminoglycosides modify the in vitro metachromatic reaction and murine generalized Shwartzman phenomenon induced by Salmonella minnesota R595 lipopolysaccharide.
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Aminoglycosides modify the in vitro metachromatic reaction and murine generalized Shwartzman phenomenon induced by Salmonella minnesota R595 lipopolysaccharide.

机译:氨基糖苷类修饰明尼苏达沙门氏菌R595脂多糖诱导的体外变色反应和鼠类广义Shwartzman现象。

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摘要

Endotoxin-neutralizing activity may be an important property for antibiotics to be used in severe sepsis. Several antibiotics, belonging to different classes, were evaluated as to their endotoxin-neutralizing ability, using the inhibition of an in vitro metachromatic assay for lipopolysaccharides and a murine generalized Shwartzman reaction model. Gentamicin, amikacin, and sisomicin have been found to share significant in vitro antiendotoxin activity at an antibiotic/endotoxin ratio as low as 1.0/5 (by weight) and to reduce the murine generalized Shwartzman reaction at an antibiotic/endotoxin ratio of 3.3/5.
机译:内毒素中和活性可能是用于严重脓毒症的抗生素的重要特性。通过抑制脂多糖的体外变色分析和鼠类广义Shwartzman反应模型,评估了几种不同类别的抗生素的内毒素中和能力。已发现庆大霉素,阿米卡星和西索米星在低至1.0 / 5(按重量计)的抗生素/内毒素比率下具有显着的体外抗内毒素活性,并在3.3 / 5的抗生素/内毒素比率下减少鼠类广义Shwartzman反应。

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